PF-06747775 (Pfizer) Third generation covalent EGFR inhibitors
Share: PF-06747775 (Pfizer) PF06747775; PF06747775; PF 06747775; PF6747775; PF 6747775; PF6747775. PFE-X775...
View Article罗西替尼 роцилетиниб روسيليتينيب Rociletinib, CO-1686. Third generation covalent...
Share: Rociletinib (CO-1686) AVL-301,CNX-419 Celgene (Originator) , Clovis Oncology N-(3-{[2-{[4-(4-acetylpiperazin-1-yl)-2-methoxyphenyl]amino}-5-...
View ArticleEGF 816 , Nazartinib
Share: EGF 816, Nazartinib EGF-816; EGFRmut-TKI EGF816 Novartis Ag innovator (R,E)-N-(7-chloro-1-(1-(4-(dimethylamino)but-2-enoyl)azepan-3-yl)-1H-benzo[d]imidazol-2-yl)-2-methylisonicotinamide...
View ArticleBMS 986120
Share:. BMS 986120 Originator Bristol-Myers Squibb Phase I Thrombosis 02 Apr 2015 Bristol-Myers Squibb plans a phase I trial in Thrombosis (In volunteers) in United Kingdom (NCT02439190) 01 Aug 2014...
View ArticlePF 06650808
Share:. PF 06650808 $PFE compound inspired by auristatins ALL DATA COMING……… /////////PF 06650808
View ArticleGDC 0853
Share: . GDC 0853 GDC-0853; RG 7845 3-[3-(hydroxymethyl)-4-[5-[[5-[(2S)-2-methyl-4-(oxetan-3- yl)piperazin-l-yl]-2-pyridyl]amino]-6-oxo-lH-pyridin-3-yl]-2-pyridyl]-7,7-dimethyl-l, 2,6,8-...
View ArticleGLPG 1690
Share: GLPG 1690 2-[[2-ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]-methylamino]-4-(4-fluorophenyl)-1,3-thiazole-5-carbonitrile $GLPG compound...
View ArticleAZD 7594
Share: . Picture credit….Bethany Halford AZD 7594 $AZN‘s asthma candidate AZ13189620; AZD-7594 Bayer Pharma Aktiengesellschaft, Astrazeneca Ab Molecular Formula: C32H32F2N4O6 Molecular Weight:...
View ArticlePF 06650833
Share: . Picture credit….Bethany Halford PF 06650833 MFC18H20FN3O4, MW361.37 1-{[(2S,3S,4S)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide...
View ArticleLY 2922470
Share: LY 2922470 as per WO2013025424A1 LY 2922470 Picture credit….Bethany Halford (3S)-3-[4-[[5-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]thiophen-2-yl]methoxy]phenyl]hex-4-ynoic acid...
View ArticleTripeptide Glycyl-L-Prolyl-L-Glutamate (Gly-Pro-Glu or GPE)
Share: Gly-Pro-Glu Synonym: GPE, Glycyl-prolyl-glutamic acid, (1-3)IGF-1 Pfizer (Originator) Neuren Pharmaceuticals (Originator) Glypromate; glycine-proline-glutamate (neuroprotectant), Neuren CAS...
View ArticleDS-1040, Activated thrombin activatable fibrinolysis (TAFIa) inhibitor
Share: DS-1040 Daiichi Sankyo Co Ltd Ischemic stroke (2S)-5-amino-2-[[1-(4-methylcyclohexyl)imidazol-4-yl]methyl]pentanoic acid 1H-Imidazole-4-propanoic acid,...
View ArticleAUNP-12 from Aurigene Discovery Technologies Limited
Share: AUNP-12 AUR-012; Aurigene-012; NP-12, Aurigene; PD-1 inhibitor peptide (cancer), Aurigene; PD-1 inhibitor peptide (cancer), Aurigene/ Pierre Fabre; W-014A Company Aurigene Discovery...
View ArticleCRD 1152, CURADEV PHARMA PRIVATE LTD
Share:Several candidates……One is …..CRD1152 ONE OF THEM IS CRD 1152 Kynurenine pathway regulators (solid tumors) Compound 2 CAS1638121-21-7 US159738837 N3-(3-Chloro-4- fluorophenyl) furo[2,3-...
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Share: MF C18H22N2O MW: 282.17321 GDC-0919; NLG-919; RG-6078, GDC0919; GDC-0919; GDC 0919; NLG919; NLG 919; NLG-919; RG6078; RG-6078; RG 6078. 1-cyclohexyl-2-(5H-imidazo[5,1-a]isoindol-5-yl)ethanol...
View ArticleCFG 920, Novartis Scientists team up with Researchers at Aurigene, Bangalore,...
Share: CFG920, Inhibitor Of Prostate Cancer With Fewer Cardiac Side Effects Cas 1260006-20-9 Novartis Target: CYP17/CYP11B2 Disease: Castration-resistant prostate cancer MF C14H13ClN4O MW: 288.0778...
View ArticleDr. Reddy’s Laboratories CEO G V Prasad has been recognized as one of India’s...
Share: Dr. Reddy’s Laboratories CEO G V Prasad has been recognized as one of India’s top 5 most valuable CEOs Read more: bit.ly/CEOsRanking...
View ArticleNovartis Molecule for functionally liver selective glucokinase activators for...
Share: 2 (R)-3-Cyclopentyl-N-(5-methoxy-thiazolo[5,4-b]pyridin-2-yl)-2-[4-(4-methyl-piperazine-1-sulfonyl)-phenyl]-propionamide...
View ArticleBTI-320 (formerly PAZ320), Soluble mannan polysaccharides from Boston...
Share: BTI-320 (formerly PAZ320) PAZ 320 Non-insulin dependent diabetes Alpha-glucosidase inhibitor; Hydrolase inhibitor; Sucrose alpha-glucosidase inhibitor Composition of chemically purified...
View ArticleBMS 919373
Share: . Bethany Halford on Twitter: “BMS-919373, from $BMS for …https://twitter.com/beth_halford/status/634105343719682048 Aug 19, 2015 – BMS–919373, from $BMS for atrial fibrillation #ACSBoston MEDI...
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